Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Adenosine 3',5'-cyclic Monophosphorothioate, Sp-Isomer, Triethylammonium Salt
A cell-permeable cAMP analog that binds cAMP-receptor proteins.
MilliporeSigma™ Calbiochem™ Ifenprodil Hemitartrate
A partial non-competitive antagonist highly selective for GluN1/N2B subtype NMDA receptors (IC50
MilliporeSigma™ Calbiochem™ VEGFR2 Kinase Inhibitor III
The VEGFR2 Kinase Inhibitor III, also referenced under CAS 204005-46-9, controls the biological activity of VEGFR2 Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ FTI-276
A highly potent and selective CAAX peptidomimetic of the carboxyl terminal of Ras proteins that inhibits farnesyl transferase (FTase) in vitro (IC50 = 500 pM).
MilliporeSigma™ Calbiochem™ O-1602
A potent agonist for the putative cannabinoid receptor, G protein-coupled receptor 55 (GPR55 receptor) (EC50 = 13)
MilliporeSigma™ Calbiochem™ 7α, 25-dihydroxycholesterol
A highly potent and specific oxysterol EBI2 (GPR183) agonist with a kd of 450 pM in a saturation binding analysis, and activates EBI2 (EC50 140 pM compared wit
MilliporeSigma™ Calbiochem™ Caspase Inhibitor, Negative Control
The Caspase Inhibitor, Negative Control, also referenced under CAS 105637-38-5, controls the biological activity of Caspase. This small molecule/inhibitor is primarily used for Cancer applications.
Tocris Bioscience™ MDNI-caged-L-glutamate
Low molecular weight, organic compound that may help regulate biological process.
Tocris Bioscience™ Galiellalactone
STAT3 inhibitor; active in vivo
Tocris Bioscience™ SEA 0400
Potent Na+/Ca2+ exchanger (NCX) inhibitor.
Tocris Bioscience™ Tocriscreen™ Kinase Inhibitor Toolbox I
Contains set of kinases for screening.
Tocris Bioscience™ BI 605906
Selective IKKβ inhibitor
Tocris Bioscience™ Tocriscreen™ Kinase Inhibitor Toolbox II
Contains set of kinases for screening.
